PUBLIKÁCIE


45. Gardiánová, M.; Slížik, L.; Koreňová, A.; Považanec, F.; Berkeš, D.: A concise synthesis of enantiomerically pure aroyl-L-alanines and dihydroaroyl-L-alanines., Chemical Papers 2013, 67, 92–100.

44. Ďuriš, A.; Daich, A.; Berkeš, D. Constrained Tetramic Acids, Homostreptopyrrolidine, and their Analogues Based on Unusual Intramolecular Wittig Olefination with Phosphorus Ylides. Synlett 2011, 1631-1637.

43.  Andrej Ďuriš, Tomáš Wiesenganger, Daniela Moravčíková, Peter Baran, Jozef Kožíšek, Adam Daich, and Dušan Berkeš Expedient and Practical Synthesis of CERT-Dependent Ceramide Trafficking Inhibitor HPA-12 and Its Analogues Org. Lett., 2011, 13 (7), 1642–1645.

42. Jakubec, P.; Berkeš, D.: „Crystallisation-induced asymmetric transformation (CIAT) for the synthesis of dipeptides containing homophenylalanine.“ Tetrahedron:Asymmetry 2010, 21, 2807-2815.
41. Jakubec, P.; Petráš P.; Duriš A.; Berkeš D.: „The first example of a crystallization-induced asymmetric transformation (CIAT) in the Mannich reaction.” Tetrahedron:Asymmetry 2010, 21, 69-74.
40. Allous, I.; Comesse, S.; Berkeš, D.; Alkyat, A.; Daich, A.: „Toward the improvement of the tandem halide displacement/amide coupling spiro-cyclization as a new route to g-lactam and pyrroloisoquinoline templates.” Tetrahedron Lett., 2009, 50, 4411-4415.
39. Vandák, D.; Berkeš, D.; Kolaroviè, A.; Marko, M.: Spôsob prípravy derivátov 4,5alfa-epoxy-6-oxomorfínanu., SK 286047 (2008).
38. Berkeš, D.; Koreòová, A.;Safáø, P.; Horváthová,H.; Prónayová, N. Indolyl substituted 4-oxobut-2-enoic acids. Synthesis and aza-Michael additions., Cent. Eur. J. Chem. 2007, 5, 688-705.
37. Berkeš, D.; Jakubec, P.; Winklerová, D.; Považanec, F.; Daich, A.: CIAT with simultaneous epimerization at two stereocenters. Synthesis of substituted b-methyl-a-homophenylalanines., Org. Biomol. Chem., 2007, 121-124.
36. Jakubec, P.; Berkeš, D.; Kolaroviè, A.; Považanec, F.: Asymmetric synthesis of aliphatic a-amino and g-hydroxy-a-amino acids. Introduction of a template for crystallization-induced asymmetric transformation (CIAT)., Synthesis 2006, 4032-4040.
35. Jakubec, P.; Berkeš, D.; Šiška, R.; Gardianová, M.; Považanec, F.: Crystallisation induced asymmetric transformation (CIAT) in the synthesis of furoylalanines and furylcarbinols., Tetrahedron: Asymmetry, 2006, 17, 1629-1637.
34. Vandák, D., Berkeš, D., Kolaroviè, A., Marko, M. Zpùsob pøípravy derivátu 4,5-a-epoxy-6-morfínanu. CZ 297571 (2006).
33. Berkes D.;Gattnar O.;Manduch M.;Varga I.;Kmetty G.;Snuparek V.;Marko M.;Michalak K.;Siska K.:Zpùsob pøípravy hydrogenhalogenidu ethylesteru kyseliny 1-metyl-4-fenyl-4-piperidin-4-karboxylové a meziprodukty k jeho provádìní.. CZ 296437 (2006).
32. Jakubec, P.; Kolaroviè, A.; Berkeš, D.: Crystallization-induced asymmetric transformations in the synthesis of active prarmaceutical substances., Materials Structure, 2005, 12, 189-191.
31. Jakubec, P.; Kolarovic, A.; Berkes, D.: Crystallization-induced asymmetric transformations in the synthesis of active prarmaceutical substances., Materials Structure, 2005, 12, 189-191.
30. Berkes, D.; Kolarovic, A.; Manduch, R.; Baran, P.; Povazanec, F.:
Crystallization-Induced Asymmetric Transformations (CIAT): Stereoconvergent Acid-Catalyzed Lactonization of Substituted 2-Amino-4-Aryl-4-Hydroxybutanoic Acids., Tetrahedron-Asymmetry, 2005, 16, 1927-1934.
29. Kolarovic, A.; Berkes, D. A.; Baran, P.; Povazanec, F.:
Crystallization-Induced Asymmetric Transformation (CIAT) With Simultaneous Epimerization at Two Stereocenters. A Short Synthesis of Conformationally Constrained Homophenylalanines.. Tetrahedron Lett., 2005, 46, 975-978.
28. Berkes D.;Gattnar O.;Manduch M.;Varga I.;Kmetty G.;Snuparek V.;Marko M.;Michalak K.;Siska K.:
Sposob pripravy hydrogenhalogenidov etylesteru kyseliny 1-metyl-4-fenyl-4-piperidin-4-karboxylovej a medziprodukty na jeho vykonavanie. SK-Pat. 2005, SK-284 526.
27. Berkes, D.; Kolarovic, A.; Raptis, R. G.; Baran, P.:
Absolute Structure Determination of (2R,1 ' S)-2-(1 '-Benzyl-2 '-Hydroxyethylamino)-4-Phenylbutanoic Acid.. J. Mol. Struct., 2004, 697, 101-107.
26. Jakubec, P.; Berkes, D. A.; Povazanec, F.:
Crystallization-Induced Asymmetric Transformation. Application to Conjugate Addition of Benzylamine to Amides of Benzoylacrylic Acid.. Tetrahedron Lett., 2004, 45, 4755-4758.
25. Safar P., Horvathova H., Korenova A., Berkes D.:
4-Heteroaryl-4-oxobutenoic acids in the synthesis of nonproteinogenic a-amino acids.. Annals of the Polish Chemical Society, 2004, 3, 76-80.
24. Safar P., Korenova A., Berkes D., Horvathova H.:
Enantiomerically pure homotryptophane derivatives.. Chem. Listy, 2004, 98, 660-661.
23. Berkes, D.; Lopuch, J.; Proksa, B.; Povazanec, F.:
Optical Resolution of Ethyl 2-(Benzylamino)-4-Oxo-4-Phenylbutanoate With Tartaric Acid - A Practical Synthesis of D-Homophenylalanine.. Chem. Pap., 2003, 57, 350-354.
22. Safar P., Berkes D., Pronayova N.:
4-(1-Benzensulfonyl-1H-pyrrol-3-yl, resp. 1H-indol-3-yl)-4-oxobut-2-enova kyselina v synteze aminokyselin.. Chem. Listy, 2003, 97, 761-762.
21. Kolarovic, A.; Berkes, D.; Baran, P.; Povazanec, F.:
Crystallization-Induced Dynamic Resolution (CIDR) and Its Application to the Synthesis of Unnatural N-Substituted Amino Acids Derived From Aroylacrylic Acids.. Tetrahedron Lett., 2001, 42, 2579-2582.
20. Berkes, D.; Kolarovic, A.; Povazanec, F.:
Stereoselective Sodium Borohydride Reduction, Catalyzed by Manganese(II) Chloride, of Gamma-Oxo-Alpha-Amino Acids. A Practical Approach to Syn-Gamma-Hydroxy-Alpha-Amino Acids.. Tetrahedron Letters, 2000, 41, 5257-5260.
19. Uher, M.; Berkes, D.:
2,5-Disubstituted S-Triazolo[3,4-b] [1,3,4]Thiadiazoles.. Chem. Pap., 1999, 53, 215-217.
18. Berkes, D.; Netchitailo, P.; Morel, J.; Decroix, B.:
Synthesis of Thieno[b]Quinolizidines and Hofmann Elimination on Methiodides Derivatives.. Synthetic Commun., 1998, 28, 949-956.
17. Berkes, D.; Povazanec, F.; Pronayova, N.:
Michael Addition in the Synthesis of Alpha-Aminoacids. Stereoselective Synthesis of Gamma-Aryl-Gamma-Hydroxy-Alpha-Aminobutanoic Acids.. Chem. Listy, 1997, 91, 659-661.
16. Kozisek, J.; Berkes, D.; Decroix, B.:
4,5,6,7,8,9-Hexahydro-10-Hydroxy-5,9-Methano-4H-Thieno[3,2-c]Azonine.. Acta Cryst., 1996, C52, 1825-1826.
15. Berkes, D.; Bar, N.; Decroix, B.:
Stereoselective Reduction of New Fused Azoninones With Bridgehead Nitrogen.. J. Heterocyclic Chem., 1995, 32, 403-405.
14. Gomory, J.; Berkes, D.; Mrazkova, J.; Perdoch, V.; Belancik, F.:
Ultrazvukovy Chemicky Reaktor Pre Laboratorne Pouzitie.. Chem. Listy, 1995, 89, 594-596.
13. Berkes, D.; Decroix, B.:
Synthese De Piperidinethienoazepinones, Methanothienoazecinone Et Etude De Leur Reduction Stereoselective.. Bull. Soc. Chim. France, 1994, 131, 989-991.
12. Safar, P.; Povazanec, F.; Zalibera, L.; Berkes, D.:
Simple Preparation of 4,5-Disubstituted -2-Cyclopentenones.. Coll. Czech. Chem. Commun., 1993, 58, 555-564.
11. Berkes, D.; Marunova, E.; Kovac, J.:
Substitution of Halogens on Furan by Hydrazines. Stable Derivatives of 5-Hydrazinofurans.. Chem. Papers, 1992, 46, 38-41.
10 . Berkes, D.; Vegh, D.; Dandarova, M.:
1-(5-Nitro-2-Furyl)-2-Propenylation of Aromatic Derivatives Under Friedel-Crafts Conditions.. Chem. Papers, 1992, 46, 333-336.
9. Uher, M.; Berkes, D.; Beno, A.:
Haloacetylisothiocyanates in the Synthesis of Fused Furans.. Acta F. R. N. Univ. Commen. - Chimia, 1992, 40, 85-91.
8. Uher, M.; Berkes, D.; Konecny, V.; Beno, A.:
Chlorinated Derivatives of N-Phenyl-N?-Chloroacetylthiourea.. Acta F. R. N. Univ. Commen. - Chimia, 1992, 40, 67-76.
7. Berkes, D.; Vegh, D.; Kovac, J.:
Sposob pripravy substituovanych 3-heteroaroyl-2,3-dibrompropanovych kyselin., 1990, CZ-Pat 260336.
6. Berkes D.;Kacina R.;Gomory J.;Frankova M.;Niznansky J.:
Sposob pripravy 1-bromdodekanu., 1990, CZ-Pat 270876.
5. Berkes, D.; Kovac, J.:
Reactions of Substituted 2-(2-Furyl)-1,2,2-Ethylnetricarbonitriles With Primary and Secondary Amines.. Chem. Papers, 1989, 43, 579-588.
4. Stasko, A.; Berkes, D.; Biskupic, S.; Pelikan, P.; Polakovic, J.:
Ion Radical of Substituted 2-Furylethenetricarbonitriles (an ESR, Quantum Chemical, and Electrochemical Study).. Chem. Papers, 1989, 43, 177-190.
3. Berkes, D.; Kovac, J.:
3-(5-halogen-2-furyl)-3-kyano-2-substituovane derivaty kyseliny propenovej a sposob ich pripravy., 1989, CZ-Pat 254207.
2. Berkes, D.; Kovac, J.:
5-Tricyanovinyl-2-Furylation of Aromatic Derivatives.. Coll. Czech. Chem. Commun., 1989, 51, 1450-1454.
1. Uher, M.; Berkes, D.; Lesko, J.; Floch, L.:
Reactions of Carbonyl Isothiocyanates With Nucleophilic Bifunctional Reagents.. Coll. Czech. Chem. Commun., 1983, 48, 1651-1658.

Výskum biotechnológií

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Spoločný projekt Biotika a.s. a STU  (ITMS 26220220093) riešený na Detašovanom pracovisku FCHPT STU Hlohovec zameraný  na výskum sekundárnych metabolitov ako enzýmových inhibítorov v metabolizme lipidov a na výskum nového postupu na prípravu vybraného enzýmového inhibítora.

Projekt je súčasťou OP Výskum a vývoj, výzvy OPVaV - 2009/2.2/03-SORO.

doba riešenia 07/2010 - 06/2014 

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